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Publications

Export 194 results:
Author Title Type [ Year(Asc)]
2015
Adachi, S.; 3rd, A. B. Cognett; Niphakis, M. J.; He, Z.; Zajdlik, A.; Denis, J. D. St.; Scully, C. C. G.; Cravatt, B. F.; Yudin, A. K. Facile Synthesis Of Borofragments And Their Evaluation In Activity-Based Protein Profiling. Chemical Communications 2015, 51 (17), 3608 - 3611.
Yudin, A. K. Macrocycles: Lessons From The Distant Past, Recent Developments, And Future Directions. Chemical Science 2015, 6 (1), 30 - 49.
Zaretsky, S.; Hickey, J. L.; Tan, J.; Pichugin, D.; Denis, M. A. St.; Ler, S.; Chung, B. K. W.; Scully, C. C. G.; Yudin, A. K. Mechanistic Investigation Of Aziridine Aldehyde-Driven Peptide Macrocyclization: The Imidoanhydride Pathway. Chemical Science 2015, 6 (10), 5446 - 5455.
Yudin, A. K. Nature’S Enzymes Tricked With Xenobiotic Oxidants. ACS Central Science 2015, 1 (2), 62 - 63.
Trinchera, P.; Corless, V. B.; Yudin, A. K. Synthesis Of Previously Inaccessible Borylated Heterocycle Motifs Using Novel Boron-Containing Amphoteric Molecules. Angewandte Chemie International Edition 2015, 54 (31), 9038 - 9041.
Zaretsky, S.; Rai, V.; Gish, G.; Forbes, M. W.; Kofler, M.; Yu, J. C. Y.; Tan, J.; Hickey, J. L.; Pawson, T.; Yudin, A. K. Twisted Amide Electrophiles Enable Cyclic Peptide Sequencing. Organic & Biomolecular Chemistry 2015, 13 (27), 7384 - 7388.
2014
He, Z.; Zajdlik, A.; Yudin, A. K. Air- And Moisture-Stable Amphoteric Molecules: Enabling Reagents In Synthesis. Accounts of Chemical Research 2014, 47 (4), 1029 - 1040.
Denis, J. D. St.; Zajdlik, A.; Tan, J.; Trinchera, P.; C. Lee, F.; He, Z.; Adachi, S.; Yudin, A. K. Boron-Containing Enamine And Enamide Linchpins In The Synthesis Of Nitrogen Heterocycles. Journal of the American Chemical Society 2014, 136 (50), 17669 - 17673.
Denis, J. D. St.; Scully, C. C. G.; C. Lee, F.; Yudin, A. K. Development Of The Direct Suzuki–Miyaura Cross-Coupling Of Primary B-Alkyl Mida-Boronates And Aryl Bromides. Organic Letters 2014, 16 (5), 1338 - 1341.
Zajdlik, A.; He, Z.; St Denis, J.; Yudin, A. Efficient Preparation Of Α-Aminoboronic Acid Derivatives Via Boroalkyl Group Migration. Synthesis 2014, 46 (04), 445 - 454.
Zaretsky, S.; Hickey, J. L.; Denis, M. A. St.; Scully, C. C. G.; Roughton, A. L.; Tantillo, D. J.; Lodewyk, M. W.; Yudin, A. K. Predicting Cyclic Peptide Chemical Shifts Using Quantum Mechanical Calculations. Tetrahedron 2014, 70 (42), 7655 - 7663.
Belding, L.; Zaretsky, S.; Rotstein, B. H.; Yudin, A. K.; Dudding, T. Shifting The Energy Landscape Of Multicomponent Reactions Using Aziridine Aldehyde Dimers: A Mechanistic Study. The Journal of Organic Chemistry 2014, 79 (20), 9465 - 9471.
White, C. J.; Hickey, J. L.; Scully, C. C. G.; Yudin, A. K. Site-Specific Integration Of Amino Acid Fragments Into Cyclic Peptides. Journal of the American Chemical Society 2014, 136 (10), 3728 - 3731.
Rotstein, B. H.; Zaretsky, S.; Rai, V.; Yudin, A. K. Small Heterocycles In Multicomponent Reactions. Chemical Reviews 2014, 114 (16), 8323 - 8359.
Treder, A. P.; Tremblay, M. - C.; Yudin, A. K.; Marsault, E. Solid-Phase Synthesis Of Piperazinones Via Disrupted Ugi Condensation. Organic Letters 2014, 16 (17), 4674 - 4677.
Zaretsky, S.; Adachi, S.; Rotstein, B. H.; Hickey, J. L.; Scully, C. C. G.; Denis, J. D. St.; Courtemanche, R.; Yu, J. C. Y.; Chung, B. K. W.; Yudin, A. K. Stereocontrolled Disruption Of The Ugi Reaction Toward The Production Of Chiral Piperazinones: Substrate Scope And Process Development. The Journal of Organic Chemistry 2014, 79 (21), 9948 - 9957.
Yudin, A. K.; Chen, G.; He, Z. Synthesis Of Functionalized 1-Azabicyclo[3.1.0]Hexanes: Studies Towards Ficellomycin And Its Analogs. HETEROCYCLES 2014, 88 (2), 1299.
He, Z.; Zajdlik, A.; Yudin, A. K. Α-Borylcarbonyl Compounds: From Transient Intermediates To Robust Building Blocks. Dalton Trans. 2014, 43 (30), 11434 - 11451.
2013
Dubovyk, I.; Watson, I. D. G.; Yudin, A. K. Achieving Control Over The Branched/linear Selectivity In Palladium-Catalyzed Allylic Amination. The Journal of Organic Chemistry 2013, 78 (4), 1559 - 1575.
Chung, B. K. W.; Hickey, J. L.; Scully, C. C. G.; Zaretsky, S.; Yudin, A. K. Bicycle Synthesis Through Peptide Macrocyclization Using Aziridine Aldehydes Followed By Late Stage Disulfide Bond Installation. MedChemComm 2013, 4 (7), 1124.
Zaretsky, S.; Scully, C. C. G.; Lough, A. J.; Yudin, A. K. Exocyclic Control Of Turn Induction In Macrocyclic Peptide Scaffolds. Chemistry - A European Journal 2013, 19 (52), 17668 - 17672.
Liew, S. K.; He, Z.; Denis, J. D. St.; Yudin, A. K. Stereocontrolled Synthesis Of 1,2- And 1,3-Diamine Building Blocks From Aziridine Aldehyde Dimers. The Journal of Organic Chemistry 2013, 78 (23), 11637 - 11645.
He, Z.; Dobrovolsky, D.; Trinchera, P.; Yudin, A. K. Synthesis Of Multisubstituted Pyridines. Organic Letters 2013, 15 (2), 334 - 337.
Zajdlik, A.; Wang, Z.; Hickey, J. L.; Aman, A.; Schimmer, A. D.; Yudin, A. K. Α-Boryl Isocyanides Enable Facile Preparation Of Bioactive Boropeptides. Angewandte Chemie 2013, 125 (32), 8569 - 8573.
2012
Rotstein, B.; Yudin, A. Aziridine-2-Carboxaldehyde Dimers Undergo Homo-Ugi 4-Component-5-Center Reactions. Synthesis 2012, 44 (18), 2851 - 2858.

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