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Export 194 results:
Author Title Type [ Year(Asc)]
2017
Kaldas, S. J.; O'Keefe, K. T. V.; Mendoza-Sanchez, R.; Yudin, A. K. Amphoteric Borylketenimines: Versatile Intermediates In The Synthesis Of Borylated Heterocycles. Chemistry - A European Journal 2017, 23 (41), 9711 - 9715.
Liew, S. K.; Holownia, A.; Diaz, D. B.; Cistrone, P. A.; Dawson, P. E.; Yudin, A. K. Borylated Oximes: Versatile Building Blocks For Organic Synthesis. Chem. Commun. 2017, 53 (81), 11237 - 11240.
Mendoza-Sanchez, R.; Corless, V. B.; Q. Nguyen, N. N.; Bergeron-Brlek, M.; Frost, J.; Adachi, S.; Tantillo, D. J.; Yudin, A. K. Cyclols Revisited: Facile Synthesis Of Medium-Sized Cyclic Peptides. Chemistry - A European Journal 2017, 23 (54), 13319 - 13322.
Tan, J.; III, A. B. Cognett; Diaz, D. B.; Lum, K. M.; Adachi, S.; Kundu, S.; Cravatt, B. F.; Yudin, A. K. Multicomponent Mapping Of Boron Chemotypes Furnishes Selective Enzyme Inhibitors. Nature Communications 2017, 8 (1).
C. Lee, F.; Holownia, A.; Bennett, J. M.; Elkins, J. M.; Denis, J. D. St.; Adachi, S.; Yudin, A. K. Oxalyl Boronates Enable Modular Synthesis Of Bioactive Imidazoles. Angewandte Chemie International Edition 2017, 56 (22), 6264 - 6267.
Zaretsky, S.; Yudin, A. K. Practical Medicinal Chemistry With Macrocyclescontemporary Macrocyclization Technologies; Marsault, E., Peterson, M. L., Eds.; John Wiley & Sons, Inc.: Hoboken, NJ, USA, 2017; pp 1 - 24.
Zaretsky, S.; Yudin, A. K. Recent Advances In The Synthesis Of Cyclic Pseudopeptides. Drug Discovery Today: Technologies 2017, 26, 3 - 10.
Belding, L.; Zaretsky, S.; Yudin, A. K.; Dudding, T. Retraction Of “A Mechanistic Model For The Aziridine Aldehyde-Driven Macrocyclization Of Peptides”. The Journal of Organic Chemistry 2017, 82 (8), 4512 - 4512.
Garrett, G. E.; Diaz, D. B.; Yudin, A. K.; Taylor, M. S. Reversible Covalent Interactions Of Β-Aminoboronic Acids With Carbohydrate Derivatives. Chemical Communications 2017, 53 (11), 1809 - 1812.
Chung, B. K. W.; White, C. J.; Yudin, A. K. Solid-Phase Synthesis, Cyclization, And Site-Specific Functionalization Of Aziridine-Containing Tetrapeptides. Nature Protocols 2017, 12 (6), 1277 - 1287.
Diaz, D. B.; Yudin, A. K. The Versatility Of Boron In Biological Target Engagement. Nature Chemistry 2017, 9 (8), 731 - 742.
Mazzeo, G.; Longhi, G.; Corless, V. B.; Zajdlik, A.; Yudin, A. K.; Abbate, S. Vibrational Circular Dichroism Unveils Chiroptical, Electrical, And Magnetic Properties Of Borylated Isocyanides And Aldehydes. European Journal of Organic Chemistry 2017, 2017 (35), 5262 - 5268.
2016
Scully, C. C. G.; White, C. J.; Yudin, A. K. The Effect Of Backbone Flexibility On Site-Selective Modification Of Macrocycles. Organic & Biomolecular Chemistry 2016, 14 (43), 10230 - 10237.
Liew, S. K.; Kaldas, S. J.; Yudin, A. K. A Linchpin Synthesis Of 6-Hydroxyceramides From Aziridine Aldehydes. Organic Letters 2016, 18 (24), 6268 - 6271.
Frost, J. R.; Scully, C. C. G.; Yudin, A. K. Oxadiazole Grafts In Peptide Macrocycles. Nature Chemistry 2016, 8 (12), 1105 - 1111.
Hickey, J. L.; Zaretsky, S.; Denis, M. A. St.; Chakka, S. Kumar; M. Morshed, M.; Scully, C. C. G.; Roughton, A. L.; Yudin, A. K. Passive Membrane Permeability Of Macrocycles Can Be Controlled By Exocyclic Amide Bonds. Journal of Medicinal Chemistry 2016, 59 (11), 5368 - 5376.
Low, K. E.; Ler, S.; Chen, K. J.; Campbell, R. L.; Hickey, J. L.; Tan, J.; Scully, C. C. G.; Davies, P. L.; Yudin, A. K.; Zaretsky, S. Rational Design Of Calpain Inhibitors Based On Calpastatin Peptidomimetics. Journal of Medicinal Chemistry 2016, 59 (11), 5403 - 5415.
Chung, B. K. W.; White, C. J.; Scully, C. C. G.; Yudin, A. K. The Reactivity And Conformational Control Of Cyclic Tetrapeptides Derived From Aziridine-Containing Amino Acids. Chemical Science 2016, 7 (11), 6662 - 6668.
Liew, S. K.; Holownia, A.; Tilley, A. J.; Carrera, E. I.; Seferos, D. S.; Yudin, A. K. A Study Of Boratriazaroles: An Underdeveloped Class Of Heterocycles. The Journal of Organic Chemistry 2016, 81 (21), 10444 - 10453.
Diaz, D. B.; Scully, C. C. G.; Liew, S. K.; Adachi, S.; Trinchera, P.; Denis, J. D. St.; Yudin, A. K. Synthesis Of Aminoboronic Acid Derivatives From Amines And Amphoteric Boryl Carbonyl Compounds. Angewandte Chemie International Edition 2016, 55 (41), 12659 - 12663.
Heine, N. B.; Kaldas, S. J.; Belding, L.; Shmatova, O.; Dudding, T.; Nenajdenko, V. G.; Studer, A.; Yudin, A. K. Synthesis Of Chiral Piperazinones Using Amphoteric Aziridine Aldehyde Dimers And Functionalized Isocyanides. The Journal of Organic Chemistry 2016, 81 (12), 5209 - 5216.
2015
Denis, J. D. St.; C. Lee, F.; Yudin, A. K. Access To Cyclic Amino Boronates Via Rhodium-Catalyzed Functionalization Of Alkyl Mida Boronates. Organic Letters 2015, 17 (23), 5764 - 5767.
Denis, J. D. St.; He, Z.; Yudin, A. K. Amphoteric Α-Boryl Aldehyde Linchpins In The Synthesis Of Heterocycles. ACS Catalysis 2015, 5 (9), 5373 - 5379.
Adachi, S.; Liew, S. K.; C. Lee, F.; Lough, A.; He, Z.; Denis, J. D. St.; Poda, G.; Yudin, A. K. Condensation-Driven Assembly Of Boron-Containing Bis(Heteroaryl) Motifs Using A Linchpin Approach. Organic Letters 2015, 17 (22), 5594 - 5597.
Chung, B. K. W.; Yudin, A. K. Disulfide-Bridged Peptide Macrobicycles From Nature. Organic & Biomolecular Chemistry 2015, 13 (33), 8768 - 8779.

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