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2017
Zaretsky, S.; Yudin, A. K. Practical Medicinal Chemistry With Macrocyclescontemporary Macrocyclization Technologies; Marsault, E., Peterson, M. L., Eds.; John Wiley & Sons, Inc.: Hoboken, NJ, USA, 2017; pp 1 - 24.
Zaretsky, S.; Yudin, A. K. Recent Advances In The Synthesis Of Cyclic Pseudopeptides. Drug Discovery Today: Technologies 2017, 26, 3 - 10.
Belding, L.; Zaretsky, S.; Yudin, A. K.; Dudding, T. Retraction Of “A Mechanistic Model For The Aziridine Aldehyde-Driven Macrocyclization Of Peptides”. The Journal of Organic Chemistry 2017, 82 (8), 4512 - 4512.
2016
Hickey, J. L.; Zaretsky, S.; Denis, M. A. St.; Chakka, S. Kumar; M. Morshed, M.; Scully, C. C. G.; Roughton, A. L.; Yudin, A. K. Passive Membrane Permeability Of Macrocycles Can Be Controlled By Exocyclic Amide Bonds. Journal of Medicinal Chemistry 2016, 59 (11), 5368 - 5376.
Low, K. E.; Ler, S.; Chen, K. J.; Campbell, R. L.; Hickey, J. L.; Tan, J.; Scully, C. C. G.; Davies, P. L.; Yudin, A. K.; Zaretsky, S. Rational Design Of Calpain Inhibitors Based On Calpastatin Peptidomimetics. Journal of Medicinal Chemistry 2016, 59 (11), 5403 - 5415.
2015
Zaretsky, S.; Hickey, J. L.; Tan, J.; Pichugin, D.; Denis, M. A. St.; Ler, S.; Chung, B. K. W.; Scully, C. C. G.; Yudin, A. K. Mechanistic Investigation Of Aziridine Aldehyde-Driven Peptide Macrocyclization: The Imidoanhydride Pathway. Chemical Science 2015, 6 (10), 5446 - 5455.
Zaretsky, S.; Rai, V.; Gish, G.; Forbes, M. W.; Kofler, M.; Yu, J. C. Y.; Tan, J.; Hickey, J. L.; Pawson, T.; Yudin, A. K. Twisted Amide Electrophiles Enable Cyclic Peptide Sequencing. Organic & Biomolecular Chemistry 2015, 13 (27), 7384 - 7388.
2014
Zaretsky, S.; Hickey, J. L.; Denis, M. A. St.; Scully, C. C. G.; Roughton, A. L.; Tantillo, D. J.; Lodewyk, M. W.; Yudin, A. K. Predicting Cyclic Peptide Chemical Shifts Using Quantum Mechanical Calculations. Tetrahedron 2014, 70 (42), 7655 - 7663.
Belding, L.; Zaretsky, S.; Rotstein, B. H.; Yudin, A. K.; Dudding, T. Shifting The Energy Landscape Of Multicomponent Reactions Using Aziridine Aldehyde Dimers: A Mechanistic Study. The Journal of Organic Chemistry 2014, 79 (20), 9465 - 9471.
Rotstein, B. H.; Zaretsky, S.; Rai, V.; Yudin, A. K. Small Heterocycles In Multicomponent Reactions. Chemical Reviews 2014, 114 (16), 8323 - 8359.
Zaretsky, S.; Adachi, S.; Rotstein, B. H.; Hickey, J. L.; Scully, C. C. G.; Denis, J. D. St.; Courtemanche, R.; Yu, J. C. Y.; Chung, B. K. W.; Yudin, A. K. Stereocontrolled Disruption Of The Ugi Reaction Toward The Production Of Chiral Piperazinones: Substrate Scope And Process Development. The Journal of Organic Chemistry 2014, 79 (21), 9948 - 9957.
2013
Chung, B. K. W.; Hickey, J. L.; Scully, C. C. G.; Zaretsky, S.; Yudin, A. K. Bicycle Synthesis Through Peptide Macrocyclization Using Aziridine Aldehydes Followed By Late Stage Disulfide Bond Installation. MedChemComm 2013, 4 (7), 1124.
Zaretsky, S.; Scully, C. C. G.; Lough, A. J.; Yudin, A. K. Exocyclic Control Of Turn Induction In Macrocyclic Peptide Scaffolds. Chemistry - A European Journal 2013, 19 (52), 17668 - 17672.
2012
Scully, C. C. G.; Rai, V.; Poda, G.; Zaretsky, S.; Burns, D. C.; R. Houliston, S.; Lou, T.; Yudin, A. K. Bending Rigid Molecular Rods: Formation Of Oligoproline Macrocycles. Chemistry - A European Journal 2012, 18 (49), 15612 - 15617.