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2018
Appavoo, S. D.; Kaji, T.; Frost, J. R.; Scully, C. C. G.; Yudin, A. K. Development Of Endocyclic Control Elements For Peptide Macrocycles. Journal of the American Chemical Society 2018, 140 (28), 8763 - 8770.
2017
Denis, J. D. St.; Liew, S. K.; Scully, C. C. G.; Yudin, A. K. Activation Of Alkynylzinc Reagents By A Hemiaminal-Driven Catalytic Microenvironment. European Journal of Organic Chemistry 2017, 2017 (2), 419 - 423.
2016
Scully, C. C. G.; White, C. J.; Yudin, A. K. The Effect Of Backbone Flexibility On Site-Selective Modification Of Macrocycles. Organic & Biomolecular Chemistry 2016, 14 (43), 10230 - 10237.
Frost, J. R.; Scully, C. C. G.; Yudin, A. K. Oxadiazole Grafts In Peptide Macrocycles. Nature Chemistry 2016, 8 (12), 1105 - 1111.
Hickey, J. L.; Zaretsky, S.; Denis, M. A. St.; Chakka, S. Kumar; M. Morshed, M.; Scully, C. C. G.; Roughton, A. L.; Yudin, A. K. Passive Membrane Permeability Of Macrocycles Can Be Controlled By Exocyclic Amide Bonds. Journal of Medicinal Chemistry 2016, 59 (11), 5368 - 5376.
Low, K. E.; Ler, S.; Chen, K. J.; Campbell, R. L.; Hickey, J. L.; Tan, J.; Scully, C. C. G.; Davies, P. L.; Yudin, A. K.; Zaretsky, S. Rational Design Of Calpain Inhibitors Based On Calpastatin Peptidomimetics. Journal of Medicinal Chemistry 2016, 59 (11), 5403 - 5415.
Chung, B. K. W.; White, C. J.; Scully, C. C. G.; Yudin, A. K. The Reactivity And Conformational Control Of Cyclic Tetrapeptides Derived From Aziridine-Containing Amino Acids. Chemical Science 2016, 7 (11), 6662 - 6668.
Diaz, D. B.; Scully, C. C. G.; Liew, S. K.; Adachi, S.; Trinchera, P.; Denis, J. D. St.; Yudin, A. K. Synthesis Of Aminoboronic Acid Derivatives From Amines And Amphoteric Boryl Carbonyl Compounds. Angewandte Chemie International Edition 2016, 55 (41), 12659 - 12663.
2015
Adachi, S.; 3rd, A. B. Cognett; Niphakis, M. J.; He, Z.; Zajdlik, A.; Denis, J. D. St.; Scully, C. C. G.; Cravatt, B. F.; Yudin, A. K. Facile Synthesis Of Borofragments And Their Evaluation In Activity-Based Protein Profiling. Chemical Communications 2015, 51 (17), 3608 - 3611.
Zaretsky, S.; Hickey, J. L.; Tan, J.; Pichugin, D.; Denis, M. A. St.; Ler, S.; Chung, B. K. W.; Scully, C. C. G.; Yudin, A. K. Mechanistic Investigation Of Aziridine Aldehyde-Driven Peptide Macrocyclization: The Imidoanhydride Pathway. Chemical Science 2015, 6 (10), 5446 - 5455.
2014
Denis, J. D. St.; Scully, C. C. G.; C. Lee, F.; Yudin, A. K. Development Of The Direct Suzuki–Miyaura Cross-Coupling Of Primary B-Alkyl Mida-Boronates And Aryl Bromides. Organic Letters 2014, 16 (5), 1338 - 1341.
White, C. J.; Hickey, J. L.; Scully, C. C. G.; Yudin, A. K. Site-Specific Integration Of Amino Acid Fragments Into Cyclic Peptides. Journal of the American Chemical Society 2014, 136 (10), 3728 - 3731.
Zaretsky, S.; Adachi, S.; Rotstein, B. H.; Hickey, J. L.; Scully, C. C. G.; Denis, J. D. St.; Courtemanche, R.; Yu, J. C. Y.; Chung, B. K. W.; Yudin, A. K. Stereocontrolled Disruption Of The Ugi Reaction Toward The Production Of Chiral Piperazinones: Substrate Scope And Process Development. The Journal of Organic Chemistry 2014, 79 (21), 9948 - 9957.
2013
Chung, B. K. W.; Hickey, J. L.; Scully, C. C. G.; Zaretsky, S.; Yudin, A. K. Bicycle Synthesis Through Peptide Macrocyclization Using Aziridine Aldehydes Followed By Late Stage Disulfide Bond Installation. MedChemComm 2013, 4 (7), 1124.
Zaretsky, S.; Scully, C. C. G.; Lough, A. J.; Yudin, A. K. Exocyclic Control Of Turn Induction In Macrocyclic Peptide Scaffolds. Chemistry - A European Journal 2013, 19 (52), 17668 - 17672.
2012
Scully, C. C. G.; Rai, V.; Poda, G.; Zaretsky, S.; Burns, D. C.; R. Houliston, S.; Lou, T.; Yudin, A. K. Bending Rigid Molecular Rods: Formation Of Oligoproline Macrocycles. Chemistry - A European Journal 2012, 18 (49), 15612 - 15617.
Roxin, Á.; Chen, J.; Scully, C. C. G.; Rotstein, B. H.; Yudin, A. K.; Zheng, G. Conformational Modulation Of In Vitro Activity Of Cyclic Rgd Peptides Via Aziridine Aldehyde-Driven Macrocyclization Chemistry. Bioconjugate Chemistry 2012, 23 (7), 1387 - 1395.