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Publications

Export 159 results:
Author Title Type [ Year(Asc)]
2019
Holownia, A.; Tien, C. - H.; Diaz, D. B.; Larson, R. T.; Yudin, A. K. Carboxyboronate: A Versatile C1-Building Block. Angewandte Chemie International Edition 2019.
Appavoo, S. D.; Huh, S.; Diaz, D. B.; Yudin, A. K. Conformational Control Of Macrocycles By Remote Structural Modification. Chem Rev 2019.
Yamaguchi, A.; Kaldas, S. J.; Appavoo, S. D.; Diaz, D. B.; Yudin, A. K. Conformationally Stable Peptide Macrocycles Assembled Using The Petasis Borono-Mannich Reaction. Chem Commun (Camb) 2019.
Tan, J.; Grouleff, J. J.; Jitkova, Y.; Diaz, D. B.; Griffith, E. C.; Shao, W.; Bogdanchikova, A. F.; Poda, G.; Schimmer, A. D.; Lee, R. E.; Yudin, A. K. De Novo Design Of Boron-Based Peptidomimetics As Potent Inhibitors Of Human Clpp In The Presence Of Human Clpx. J Med Chem 2019, 62 (13), 6377-6390.
Smolyar, I. V.; Yudin, A. K.; Nenajdenko, V. G. Heteroaryl Rings In Peptide Macrocycles. Chem Rev 2019.
Mader, P.; Mendoza-Sanchez, R.; Iqbal, A.; Dong, A.; Dobrovetsky, E.; Corless, V. B.; Liew, S. K.; Houliston, S. R.; De Freitas, R. Ferreira; Smil, D.; Sena, C. C. Dela; Kennedy, S.; Diaz, D. B.; Wu, H.; Dombrovski, L.; Allali-Hassani, A.; Min, J.; Schapira, M.; Vedadi, M.; Brown, P. J.; Santhakumar, V.; Yudin, A. K.; Arrowsmith, C. H. Identification And Characterization Of The First Fragment Hits For Setdb1 Tudor Domain. Bioorg Med Chem 2019, 27 (17), 3866-3878.
Trudel, V.; Yudin, A. K. Nucleophilic Boron Clusters Lead To New Borylation Methods. Chem 2019.
Kaldas, S.; Kran, E.; Mück-Lichtenfeld, C.; Yudin, A.; Studer, A. Reaction Of Vinylaziridines With Arynes: Synthesis Of Benzazepines And Branched Allyl Fluorides. Chemistry – A European Journal 2019.
Soor, H. S.; Hansen, J.; Diaz, D. B.; Appavoo, S.; Yudin, A. K. Solid-Phase Synthesis Of Peptide Β-Aminoboronic Acids. Peptide Science 2019, 111 (1), e24072.
2017
Shao, W.; Kaldas, S. J.; Yudin, A. K. 3-Cyanoallyl Boronates Are Versatile Building Blocks In The Synthesis Of Polysubstituted Thiophenes. Chemical Science 2017, 8 (6), 4431 - 4436.
Denis, J. D. St.; Liew, S. K.; Scully, C. C. G.; Yudin, A. K. Activation Of Alkynylzinc Reagents By A Hemiaminal-Driven Catalytic Microenvironment. European Journal of Organic Chemistry 2017, 2017 (2), 419 - 423.
Kaldas, S. J.; O'Keefe, K. T. V.; Mendoza-Sanchez, R.; Yudin, A. K. Amphoteric Borylketenimines: Versatile Intermediates In The Synthesis Of Borylated Heterocycles. Chemistry - A European Journal 2017, 23 (41), 9711 - 9715.
Liew, S. K.; Holownia, A.; Diaz, D. B.; Cistrone, P. A.; Dawson, P. E.; Yudin, A. K. Borylated Oximes: Versatile Building Blocks For Organic Synthesis. Chem. Commun. 2017, 53 (81), 11237 - 11240.
Mendoza-Sanchez, R.; Corless, V. B.; Q. Nguyen, N. N.; Bergeron-Brlek, M.; Frost, J.; Adachi, S.; Tantillo, D. J.; Yudin, A. K. Cyclols Revisited: Facile Synthesis Of Medium-Sized Cyclic Peptides. Chemistry - A European Journal 2017, 23 (54), 13319 - 13322.
Tan, J.; III, A. B. Cognett; Diaz, D. B.; Lum, K. M.; Adachi, S.; Kundu, S.; Cravatt, B. F.; Yudin, A. K. Multicomponent Mapping Of Boron Chemotypes Furnishes Selective Enzyme Inhibitors. Nature Communications 2017, 8 (1).
C. Lee, F.; Holownia, A.; Bennett, J. M.; Elkins, J. M.; Denis, J. D. St.; Adachi, S.; Yudin, A. K. Oxalyl Boronates Enable Modular Synthesis Of Bioactive Imidazoles. Angewandte Chemie International Edition 2017, 56 (22), 6264 - 6267.
Zaretsky, S.; Yudin, A. K. Practical Medicinal Chemistry With Macrocyclescontemporary Macrocyclization Technologies; Marsault, E., Peterson, M. L., Eds.; John Wiley & Sons, Inc.: Hoboken, NJ, USA, 2017; pp 1 - 24.
Zaretsky, S.; Yudin, A. K. Recent Advances In The Synthesis Of Cyclic Pseudopeptides. Drug Discovery Today: Technologies 2017, 26, 3 - 10.

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